RHIF CAS Amhuredd N-Boc Sitagliptin.486460-23-5

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RHIF CAS Amhuredd N-Boc Sitagliptin.486460-23-5
Manylion
MF:C21H23F6N5O3
MW: 507.43
EINECS:1312995-182-4
Dosbarthiad cynnyrch
Canolradd Sitagliptin
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Amhuredd Sitagliptin N-Boc Gwybodaeth sylfaenol
Enw Cynnyrch: Amhuredd N-Boc Sitagliptin
Cyfystyron: Amhuredd N-Boc Sitagliptin;Boc-Sitagliptin;tert-Butyl N-[(2R)-4-oxo-4-[3-(trifluoromethyl)-6,8- dihydro-5H-[1,2,4]triazolo[4,3-a]pyrasin-7-yl]-1-(2,4,5-trifflworoffenyl )butan-2-yl]carbamad;Sitagliptin N-Boc;N-Boc-Sitagliptin;(R)-tert-Butyl (4-oxo-4-(3-(trifluoromethyl)) -5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)-1-(2 ,4,5-trifluorophenyl)butan-2-yl)carbamate;tert-butyl (R)-(4-oxo-4-(3-(trifluoromethyl)){{ 52}},6-dihydro-[1,2,4] triazolo[4,3-a]pyrazin-7(8H)-yl)-1-(2,4 ,5-trifluorophenyl)butan- 2-yl)carbamad;Amhuredd Sitagliptin 56
CAS: 486460-23-5
MF: C21H23F6N5O3
MW: 507.43
EINECS: 1312995-182-4

 

Priodweddau Cemegol Amhuredd N-Boc Sitagliptin

Ymdoddbwynt 188-191 gradd (Datrys: toluene (108-88-3))
dwysedd 1.46±0.1 g/cm3(Rhagweld)
tymheredd storio. Oergell
hydoddedd Clorofform (Ychydig, Wedi'i Gynhesu), DMSO (Ychydig), Asetad Ethyl (Ychydig)
ffurf Solet
pka 11.60±0.46(Rhagweld)
lliw Gwyn

 

Defnydd A Synthesis Amhuredd N-Boc Sitagliptin

Defnyddiau N-Boc-Sitagliptin yw deilliad gwarchodedig N-Boc o Sitagliptin (S490990), atalydd dipeptidyl peptidase-4 a ddefnyddir ar gyfer rheolaeth glycemig ar gyfer cleifion â diabetes math 2.

 

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